3-Triazole相关论文
One-Pot Synthesis of Novel 1,2,3-Triazole Containing Bisphosphonates via the Controlled Michael-Type
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Glucosamine-6 phosphate synthase(GlmS)is the first enzyme of the hexosamine biosynthetic pathway.This enzyme catalyzes t......
As a pivotal factor in the signal transduction pathways,protein tyrosine kinases(PTKs)is highly related with the oncolog......
1,2,3-Triazoles are an important class of heterocyclic compounds.They are shown to have different biological activities,......
we have developed a novel type of N2-selective coupling reaction of 1,2,3-triazoles with indole/pyrrole through a N-iodo......
Hiv-1 整合酶是抗艾滋病药物的重要作用靶点,芳基二酮酸类化合物被认为是最有效的Hiv-1 整合酶抑制剂 [1,2]。在前期发现1,2,3-三......
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Nitrogen-containing bisphosphonic acids and their salts (N-BP) represent an important class of phosphorus compounds poss......
Design,synthesis and in vitro biological evaluation of short-chain C12-sphinganine and its 1,2,3-tri
In the present study,we report the synthesis of short-chain C12-sphinganine and a small library of its 1,2,3-triazoles f......
Highly Efficient Blue Phosphorescent Organic Light-Emitting Diodes Hosted by Asymmetric Design of Bi
The intrinsic asymmetry of 1,2,3-triazole as the core was designed and synthesized three isomers,1,2 dDPAmTAz,dTPAmTAZ,a......
Synthesis and characterization of glycosyl 1,2,3-triazole anticancer compounds with hepatic targetin
Since the galactose residues can be recognized by asialoglycoprotein recepter(ASGPR)located in the mammal liver cell sur......
Synthesis,Crystal Structure and Its Application in Living Cells Imaging of Benz(c)acridine-1,2,3-tri
A highly selective iron ions fluorescent probe based on the benz(c)acridine-1,2,3-triazole derivatives was produced by m......
Synthesis,Antimicrobial Activity,and Molecular Docking of Benzoic Hydrazide or Amide Derivatives Con
Main observation and conclusionrnThe present study was carried out in an attempt to synthesize a new class of antimicrob......
Efficient Synthesis of Unnatural Amino Acids Through C(sp3)-H Activation with 1,2,3-Triazole as Easy
Unnatural amino acids are key structural motifs of peptidomimetics,peptides and many other pharmaceutically compound......
Fluorescence active fused-triazole was developed as a ligand in gold(I) cation coordination. The coordination ability wa......
报道了4-取代-1-磺酰基-1,2,3-三氮唑在绿色溶剂中的催化水解反应,以1 mol%硫酸铜作为催化剂,在水/PEG-400混合溶剂中以较高的收率......
通过使用简单的Et3N催化容易获得的β-取代NH-烯胺酯和对甲苯磺酰叠氮的反应,高效实现了全取代的1,2,3-三氮唑的合成.在该方法中,......
目的 设计合成一系列司他夫定类衍生物,并评价其抗肿瘤活性.方法 以司他夫定为原料,经磺酸酯化后与叠氮化钠反应生成5'-叠氮基司他......
目的 设计合成一系列新型1,2,3-三氮唑类化合物,评价其抗人类巨细胞病毒和带状疱疹病毒活性.方法 氰基乙酸乙酯与叠氮化物进行环加......
Synthesis and Crystal Structure of 2-P-Methyloxyphenyl-3a-(2-phenyl-1,2,3-triazole-4-yl)-3,4-dihydro
本文通过对荣华二采区10...
本文通过对荣华二采区10...
以1-氨基-1,2,3-三唑(1)为原料,经二氯异氰尿酸钠(SDCI)氧化偶联合成了具有稳定N8结构(8个氮原子直接相连)和光致变色特性的新型多......
A Double Azole-bridged Dinuclear Copper(Ⅱ) Complex Containing 4-Pyridyl-NH-1,2,3-triazoles:Synthesis
A new dinuclear copper(Ⅱ) compound[Cu2(CH3COO)2(L)2(H20)2]·4H20 (1,HL =4-pyridyl-NH-1,2,3-triazole) has been synthesiz......
Synthesis and Crystal Structure of a Dinuclear Cu(Ⅱ) Complex Based on a Carboxyl-substituted 1H-1,2,
The novel dinuclear copper complex [Cu2(H2O)2(DMF)2(L)2](1, H2 L = 5-phenyl-2H-1,2,3-triazole-4-carboxylic acid, DMF = N......
Synthesis and Antibacterial Activities of 1,4-Disubstituted Phenyl-5-(halo-2-hydroxyphenyl)imino-1,2
本文通过对荣华二采区10...
Synthesis and Biological Activities of Novel Thiophosphoryl Oximates Containing Thiazole and 1,2,3-T
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
Synthesis,Characterization and Thermal Behaviors of 4-Amino-5-nitro-1,2,3-triazole(ANTZ)and Its Deri
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
Facile Synthesis of 4,5-Disubstituted 2H-1,2,3-Triazoles by Catalyst-free Cycloaddition between Subs
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
Cyclometalated Ruthenium Complexes of 1,2,3-Triazole-containing Ligands: Synthesis, Structural Studi
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
Synthesis and Insecticidal Evaluation of Novel Phthalic Diamides Containing 1,2,3-Triazoles via Clic
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
Synthesis and Antibacterial Activities of 1,4-Disubstituted Phenyl-5-(halo-2-hydroxyphenyl)imino-1,2
According to the superposition principle af reinforcement of biological activities,24 novel 1,4-disubstituted phenyl-5-(......
1H-1,2,3-三唑类化合物是一类重要的杂环化合物,由于其独特的化学性质和生物活性,在医药、农药和工业方面都得到广泛的应用。本文......
利用CuI/NBS这种新型催化体系来促进单-6-叠氮-β-环糊精与苯乙炔之间的偶联反应,通过这个多组分反应可以高效地以炔和叠氮为原料......
以2-苯基-1,2,3-三唑-4-甲酸为原料,经酰氯化,得到2-苯基-1,2,3-三唑-4-甲酰氯,在PEG-400为相转移催化剂的条件下,与硫氰酸铵及酰......
采用对甲苯磺酸催化合成N1-烷基-1,2,3-三氮唑和N2-烷基-1,2,3-三氮唑。两种产物均有紫外吸收，但只有N2-烷基-1,2,3-三氮唑有荧光。......
研究5-烷氧-3,4-二溴-2（5H）-呋喃酮与末端炔烃、叠氮化钠的＂一锅煮＂反应,没有得到预期的稠杂环化合物,仅得到了5-烷氧-4-三唑基-3-溴2（5......
以对氯氯苄为原料，经取代、I，3-偶极环加成和缩合反应得到含1，2，3-三唑环的α，γ-二酮衍生物，其结构经1HNMR,13CNMR以及Ms确证。研究表明......
在微波辐射、无溶剂、无催化条件下,合成了两个新型含1,2,3-三唑基的α-氨基膦酸酯类化合物,结构经IR、NMR、X-射线晶体衍射进行了......
本文研究1-芳基-4-乙氧羰基-5-氨基-1,2,3,-连三唑(1)同过量乙酸,乙酸酐、乙酰氯、苯甲酰氯以及甲酰胺等的反应,制得1的14种新衍生......
1,2,3-三唑(1)可广泛用于杀菌剂、杀虫剂的制备,亦可用于合成他唑巴坦(tazobactam)等β-内酰胺类抗生素[1],在高分子化工中也有重......
期刊
用密度泛函B3LYP/6-311＋＋G＊＊方法,对气相和水相中的5-醛基-1,2,3-三唑互变异构体进行了几何构型全自由度优化,获得了它们在气相和水相......
开展了2,3,4,6-四-O-特戊酰基-β-D-吡喃葡萄糖叠氮与炔烃的1,3-偶极环加成反应的研究,并首次合成了一种新的1-（2,3,4,6-四-O-特戊......
以4-氨基-3-（4-甲基-1,2,3-噻二唑）-1,2,4-三唑-5-硫酮为原料,与醛在冰乙酸中回流制得15个新型4-取代亚氨基-3-（4-甲基-1,2,3-噻二唑）-......
设计并合成了15个未曾见文献报道的1-（2-（4-取代）苯氧乙基）-1H-1,2,3-三氮唑衍生物,并通过NMR、IR、MS确认了它们的结构.对合成条件进......
以1,1′-联-2-萘酚为原料,经过丙炔化成醚反应和两次Click反应,制备了两个不对称双-1,2,3-三氮唑类化合物A和B,用1H NMR和13C NMR......
本文报道了用D-阿拉伯-己醛糖脎合成糖接三唑的基本方法,并由此合成了一系列接三唑衍生物,元素分析、<sup>1</sup>H-NMR,<sup>13</......
